Question:

Non-linear pharmacokinetics is most likely due to _____.

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Saturation of enzymes → metabolism can't keep up → non-linear kinetics.
Updated On: Jun 16, 2025
  • first-pass metabolism
  • saturation of metabolic enzymes
  • renal excretion
  • high plasma protein binding
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The Correct Option is B

Solution and Explanation

Non-linear pharmacokinetics often arises when drug concentrations saturate enzymes responsible for metabolism, resulting in a disproportionate increase in drug levels with dose.
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